Latest update


Last approved inhibitor(s)

Pexidartinib, Entrectinib, Fedratinib, Upadacitinib, Alpelisib

New inhibitor(s) this month

Ceralasertib, Derazantinib, Lazertinib, Pralsetinib, Ripretinib, Rivoceranib, Samotolisib


Structures and data are compiled by SB&C Team from the Chembl Drugstore and
Please note that we provide information about inhibitors having known International Nonproprietary Names (INN). For more information see the USAN nomenclature.


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How to cite PKIDB

Carles, F., Bourg, S., Meyer, C., and Bonnet, P. (2018). PKIDB: A Curated, Annotated and Updated Database of Protein Kinase Inhibitors in Clinical Trials. Molecules 23, 908. DOI: 10.3390/molecules23040908